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Found 3 of ic50 data for polymerid = 49000987,50002151,50006935,50007539
TargetP2X purinoceptor(Macaca mulatta)
Janssen Research And Development

Curated by ChEMBL
LigandPNGBDBM254266(US10112937, Example 158 | US10150765, Example 158 ...)
Affinity DataIC50:  7.90nMAssay Description:Antagonist activity at macaque P2X7 assessed as inhibition of BzATP-induced calcium flux preincubated for 30 mins followed by BzATP addition measured...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor(Cavia porcellus)
University Of Leeds

Curated by ChEMBL
LigandPNGBDBM50087267((1-(N,O-bis(1,5-isoquinolinesulfonyl)-N-methyl-L-t...)
Affinity DataIC50:  130nMAssay Description:Inhibition of guinea pig P2X7 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor(Mus musculus)
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM85043(CAS_149017-66-3 | CHEMBL69234 | NSC_6093163 | PPAD...)
Affinity DataIC50:  2.10E+4nMAssay Description:Inhibition of inward ion current elicited by ATP at mouse P2X4 receptor (mutant type)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed